ʻO ka hoʻokomo ʻana i ka Citrus Aurantium Extract

ʻO ka hoʻokomo ʻana i ka Citrus Aurantium

Citrus Aurantium, he mea kanu no ka ohana rutaceae, ua laha nui ia ma Kina.ʻO Citrus aurantium ka inoa Kina no ka lime.I ka lāʻau lapaʻau kuʻuna Kina, ʻo citrus aurantium kahi lāʻau kuʻuna kanaka i hoʻohana nui ʻia e hoʻonui i ka ʻai a hoʻoponopono i ka qi (ikaika).Ma Italia, ʻo ka citrus aurantium kekahi lāʻau lapaʻau kuʻuna mai ka makahiki 16, i hoʻohana ʻia e mālama i ke kuni e like me ka maʻi maʻi maʻi a ma ke ʻano he antimicrobial agent.Ua hōʻike ʻia nā haʻawina hou e hiki ai i ka citrus aurantium ke pani i ka ephedra i ka mālama ʻana i ka momona me ka ʻole o nā hopena ʻaoʻao cardiovascular.

ʻO ka mea waiwai o ka citrus aurantium he hesperidin, neohesperidin, nobiletin, auranetin, aurantiamarin, nuringin, synephrine, limonin.

ʻO Citrus Aurantium Extract-Ruiwo

 

Mea hoʻoikaika kino

hesperidin, neohesperidin, nobiletin, D-limonene, auranetin, aurantiamarin, citrin, synephrine, limonin

Waiwai kino

Crystallization, helu heheʻe 184-1850C, carbonate crystallization 151-152, hiki ke hoʻoheheʻe ʻia i ka wai.Bitartrate, wahi hehee 188-189, hiki ke hooheheeia iloko o ka wai, paakiki e hemo i ka ethanol, aneane hiki ole ke hooheheeia iloko o ka chloroform, etera.Hydrochloride, aniani kala ʻole (ethanol-ethyl ether), helu heheʻe 166-167.He mea maʻalahi ka racemization i ka hoʻokaʻawale chromatography o ka waika ikaika a me ka resin exchange ion base.

Ka hopena lāʻau lapaʻau
1. Ka hopena ma ka ʻōpū: Fructus Aurantii a me Fructus Aurantii Fructus Decoction mai ʻekolu mau wahi hana like ʻole (Sichuan, Jiangxi, a me Hunan) i hōʻike i kahi hopena pale i ka ʻōpū in vitro o nā ʻiole (hāpai a ʻaʻole hāpai);Ua hauʻoli ka ʻōpū o ka lapeti i loko o ka vivo a me ka in vitro (hāpai a ʻaʻole hāpai).Ua hōʻike pū ʻia ka fistula uterine rabbit i ka hoʻoikaika ʻana i ka ʻōpū o ka ʻōpū, ka hoʻonui ʻana i ka haʻalulu, a me ka hoʻopaʻapaʻa tetanic.Hiki i ka Fructus Aurantii tincture a me ka Fructus Aurantii wai extract ke hoʻoulu i ka ʻōpū rabbit (in vivo a in vitro).Kāohi ʻia ka ʻōpū ʻiole (in vitro).ʻO kahi mea alkaloid i hoʻokaʻawale ʻia mai Fructus Aurantii a me Lycium ʻalani kekahi i loaʻa kekahi hopena contractile i ka ʻōpū o ka rabbit in vitro, ʻoi aku hoʻi ma ka ʻiʻo ʻōpū i hoʻoulu ʻia e ka pituitrin.ʻO ka ʻāpana o ka alkaloid i wehe ʻia he hopena hoʻomaha i ka ʻōpū o ka rabbit in vitro, a ʻoi aku ka ʻike o ka hopena hoʻomaha o ka ʻōpū ma hope o ka hypophysial excitation.ʻO Cirantin, i hoʻokaʻawale ʻia mai Fructus Aurantii Fructus Peel, ke kāohi i ka hana hyaluronate a puni ka ovary, e pili ana paha i kona hopena contraceptive (pale i ka fertilization).

2. Ka hopena ma ka ʻōpū: ʻO Fructus Aurantii a me Fructus Aurantii mai nā wahi ʻokoʻa ʻekolu i kāohi i ka ʻōpū i nā ʻiole a me nā rapeti;Ua pāpā ʻia ka hapa nui o nā ʻōpū ʻōpū o ka lapeti, akā ʻaʻohe mea i loli.Ua kāohi ʻo Fructus Aurantii a me kāna mea hoʻoheheʻe wai i nā paipu ʻōpū o nā ʻiole (in vitro) a me nā lākeke (in vitro).ʻO ke kiʻekiʻe kiʻekiʻe (1: 1000) i kāohi i ka'ōpū liʻiliʻi o nā lapeti i hoʻokaʻawaleʻia a me nā puaʻa puaʻa a pale i nā hopena o ka acetylcholine a me ka histamine.ʻO ka haʻahaʻa haʻahaʻa (1: 10 000), ma hope o kahi manawa pōkole o ka inhibition, hiki ke hōʻike i kahi hopena excitatory, hoʻonui amplitude, a me ka wikiwiki.I nā ʻīlio anesthetized, ua pāpā ʻia ke alo o ka ʻōpū e nā decoctions.Akā no nā ʻīlio me ka gastroenterostomy, loaʻa iā ia kahi hopena hoʻonāukiuki, hiki ke hoʻoikaika i ka neʻe ʻana o ka ʻōpū a me ke kani ʻana.

3. Nā hopena ma ka puʻuwai a me nā kīʻaha koko: ka liʻiliʻi o ka excitability a me ka nui o ka inhibition ma ka puʻuwai o ka toad in vitro.Fructus Aurantii a me Fructus Aurantii Aurantii aqueous decoction, Fructus Aurantii tincture, a me ka wai extract ua like.ʻO ka decoction Fructus Aurantii a i ʻole ka waiʻona i hoʻopaʻa ʻia i loko o ke kino hiki ke hopena i ka hoʻonui nui ʻana i ka pressor.Ua hōʻike ʻia ʻo Fructus Aurantii a me Fructus Aurantii Fructus mai ʻekolu mau wahi noho like ʻole he hopena vasoconstriction ma ke kino holoʻokoʻa.I nā ʻīlio anesthetized, aia kahi hopena koʻikoʻi a wikiwiki hoʻi.ʻAʻohe ʻeha hanu a i ʻole hypotension i hoʻokumu ʻia e ka epinephrine, a ʻaʻohe piʻi aʻe o ka puʻuwai.

ʻO ka mīkini hoʻoikaika ikaika e pili ana i nā kumu penei:

3.1.ʻO ka hauʻoli o nā mea loaʻa α, e hoʻoulu ai i ka vasoconstriction i kekahi mau ʻāpana (hiki i ka phenylzoline ke hoʻohuli i ka hoʻonui ʻana i ke kaomi i kahi hopena antihypertensive).

3.2.Hoʻonui ʻia ka hoʻopaʻa ʻana o ka myocardial a me ka hoʻonui ʻana i ka puʻuwai puʻuwai (isolated guinea pig heart perfusion and cardiopulmonary preparation).Ma hope o ka reserpine, ʻoi aku ka koʻikoʻi o ka hopena hoʻoikaika ikaika o Fructus aurantii aurantii.Ua hoʻonui nui ʻia ke kahe o ke aʻa coronary (289.4% ka piʻi ʻana o ke aʻaʻa coronary e ka bubble flowmeter) a me ka hoʻonui ʻana i ke kahe o ke koko a me ka lolo e 86.4% a me 64.5% ma ka awelika, he ʻokoʻa loa ia mai ka norepinephrine.Ua emi iho ke kahe o ke koko femoral a me ka hoʻonui iki ʻana i ka hoʻohana ʻana o ka oxygen myocardial, ʻaʻole i kūlike me ka piʻi nui o ke kahe coronary.Ma nā ho'āʻo ECG i nā ʻīlio a me nā puaʻa guinea, ʻaʻole koʻikoʻi ka arrhythmia (ventricular tachycardia a i ʻole atrioventricular block) ma muli o ka nui o ka aurantii aurantii.Ma muli o nā hiʻohiʻona i luna, ua ʻōlelo ʻia e mālama i ka haʻalulu cardiogenic.Hiki i nā Alkaloids i hoʻokaʻawale ʻia mai Fructus Aurantii a me Lycium ʻalani hiki ke hoʻoikaika i ka ʻāʻī o ka ʻiʻo maʻemaʻe vascular, ʻoi aku ke mālama ʻia me ka pituitrin.

4. Antithrombotic: In vitro ho'āʻo o 0.1g/ml Fructus Aurantii aqua decoction hōʻike i ka maopopo antithrombotic hopena.

5. Anti-allergic reaction: 100mg/kg static pulse injection o Fructus Aurantii Aurantii wai extract hiki ke inhibit passive ili allergic reaction (PCA) i na iole, a me 50μg/ml hiki inhibit histamine hookuu mai iole abdominal mast pūnaewele.

6. Nā hopena ʻē aʻe: Hiki i ka citrus plant mycin ke hoʻemi i ka ʻike o ka cholestatin i loko o ka serum a me ke akepaʻa o nā ʻiole i hānai ʻia me ka meaʻai cholesterol.He hopena pale ka waiʻona o Fructus Aurantii i ka mycobacterium tuberculosis H37Rv in vitro, a he 1:1000 kona hoʻokuʻu ʻana.ʻAʻohe hopena o kāna decoction wai i ka bronchus puaʻa guinea.Ua hōʻike ʻia ʻo ka wai hua citrus e hoʻonui i ka helu fermentation o ka hū a ʻaʻole e hoʻemi i kāna hana ma hope o ka hoʻolapalapa ʻana, no laila ʻaʻole ia he mea enzymatic.ʻO ka hoʻohana lapaʻau nui o ka wai ʻalani, ʻo ia ka waiwai o ka huaora C a loaʻa iā ia ka nui o nā huaora A a me B. ʻAʻole i loko o ka ʻili ka huaora C akā waiwai i ka huaʻa A. He ʻawaʻawa a hiki ke hoʻoikaika i ka ʻōpū.Hiki i nā keiki e like me ka lawe ʻana i ka nui o nā peels ke hoʻoulu i ka ʻona (ʻeha ʻōpū, ʻāʻī).

Kuhi: http://www.a-hospital.com

No ka meaʻO Citrus Aurantium Extract, e ʻoluʻolu e kelepona mai iā mākou.Ke kali nei mākou iā ʻoe ma ʻaneʻi i kēlā me kēia manawa!!!

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Ka manawa hoʻouna: Dec-15-2022