ʻO ka hoʻolauna ʻana o Citrus Aurantium
ʻAurantium Citrus, he mea kanu no ka ʻohana rutaceae, ua hoʻolaha nui ʻia ma Kina. ʻO Citrus aurantium ka inoa kuʻuna Kina no ka lime. I ka lāʻau lapaʻau kuʻuna Kina, ʻo ka citrus aurantium kahi lau nahele kuʻuna i hoʻohana nui ʻia e hoʻonui i ka makemake a hoʻoponopono i ka qi (ikehu). Ma Italia, ʻo ka citrus aurantium kekahi lāʻau lapaʻau kuʻuna mai ke kenekulia 16, i hoʻohana ʻia e mālama i ke kuni e like me ka malaria a ma ke ʻano he mea antimicrobial. Ua hōʻike ʻia nā haʻawina hou e hiki i ka citrus aurantium ke pani i ka ephedra i ka mālama ʻana i ka momona me ka ʻole o nā hopena ʻino o ka cardiovascular.
ʻO nā ʻāpana kūpono o ka citrus aurantium he hesperidin, neohesperidin, nobiletin, auranetin, aurantiamarin, nuringin, synephrine, limonin.
Mea hana nui
hesperidin, neohesperidin, nobiletin, D-limonene, auranetin, aurantiamarin, citrin, synephrine, limonin
Waiwai kino
ʻO ke kristal ʻana, ka wahi hoʻoheheʻe 184-1850C, ke kristal ʻana o ka carbonate 151-152, maʻalahi ka hoʻoheheʻe ʻana i ka wai. Bitartrate, wahi hoʻoheheʻe 188-189, hiki ke hoʻoheheʻe ʻia i ka wai, paʻakikī ke hoʻoheheʻe ʻia i loko o ka ethanol, aneane hiki ʻole ke hoʻoheheʻe ʻia i loko o ka chloroform, ether. Hydrochloride, kristal kala ʻole (ethanol-ethyl ether), wahi hoʻoheheʻe 166-167. He maʻalahi ka racemization e hana i ka hoʻokaʻawale ʻana o ka chromatography o nā resins hoʻololi ion waikawa ikaika a me ke kumu.
Ka hopena lāʻau lapaʻau
1. Hopena ma ka ʻōpū: Ua hōʻike ʻo Fructus Aurantii a me Fructus Aurantii Fructus Decoction mai ʻekolu mau wahi hana like ʻole (Sichuan, Jiangxi, a me Hunan) i kahi hopena pale ma ka ʻōpū in vitro o nā ʻiole (hāpai a me ka hāpai ʻole); Ua hoʻonāukiuki ʻia ka ʻōpū rabbit i loko o ke kino a me ka in vitro (hāpai a ʻaʻole hāpai). Ua hōʻoia pū ka fistula uterine rabbit e hoʻoikaika i nā ʻūlū ʻōpū, hoʻonui i ke kaumaha, a me ka ʻūlū tetanic. Hiki i ka tincture Fructus Aurantii a me ka wai Fructus Aurantii ke hoʻonāukiuki i ka ʻōpū rabbit (in vivo a me in vitro). Ua kāohi ʻia ka ʻōpū ʻiole (in vitro). Loaʻa i kahi mea alkaloid i hoʻokaʻawale ʻia mai Fructus Aurantii a me Lycium orange kahi hopena contractile i ka ʻōpū rabbit i loko o ke kino, ʻoi aku hoʻi ma ka ʻiʻo uterine i hoʻonāukiuki ʻia e ka pituitrin. ʻO ka ʻāpana o ka alkaloid i wehe ʻia he hopena hoʻomaha ma ka ʻōpū rabbit i loko o ke kino, a ʻoi aku ka maopopo o ka hopena hoʻomaha o ka ʻōpū ma hope o ka hoʻonāukiuki hypophysial. ʻO Cirantin, i hoʻokaʻawale ʻia mai Fructus Aurantii Fructus Peel, kāohi i ka hana hyaluronate a puni ka ovary, kahi e pili ana paha i kona hopena contraceptive (e pale ana i ka fertilization).
2. Hopena ma ka ʻōpū: ʻO Fructus Aurantii lāua ʻo Fructus Aurantii mai ʻekolu mau wahi noho like ʻole i kāohi i ka ʻōpū i loko o nā ʻiole a me nā lāpaki; Ua kāohi ʻia ka hapa nui o nā ʻōpū ʻōpū i loko o nā lāpaki, akā ʻaʻohe loli iki. Ua kāohi ʻo Fructus Aurantii a me kāna wai wai i nā ʻōpū ʻōpū o nā ʻiole (in vitro) a me nā lāpaki (in vitro). ʻO ke kiʻekiʻe o ka noʻonoʻo (1:1000) i kāohi i ka ʻōpū liʻiliʻi o nā lāpaki i hoʻokaʻawale ʻia a me nā puaʻa guinea a kāohi i nā hopena o ka acetylcholine a me ka histamine. ʻO ka noʻonoʻo haʻahaʻa (1:10 000), ma hope o kahi manawa pōkole o ke kāohi ʻana, hiki ke hōʻike i kahi hopena hoʻonāukiuki, hoʻonui ʻia ka amplitude, a hoʻolalelale ʻia ke alapine. I nā ʻīlio anesthetized, ua kāohi maopopo ʻia ke alo o ka ʻōpū e nā decoctions. Akā no nā ʻīlio me ka gastroenterostomy, loaʻa iā ia kahi hopena hoʻonāukiuki, hiki ke hoʻoikaika i ka neʻe ʻana o ka gastrointestinal a me ke ʻano o ka contraction.
3. Nā hopena ma ka puʻuwai a me nā kīʻaha koko: ka liʻiliʻi o ka hoʻonāukiuki a me ka nui o ka pale ʻana ma ka puʻuwai o ka toad in vitro. ʻO ka wai hoʻoheheʻe ʻo Fructus Aurantii a me Fructus Aurantii Aurantii, ka tincture Fructus Aurantii, a me ka wai hoʻokahe like. ʻO ka hoʻoheheʻe ʻana o Fructus Aurantii a i ʻole ka wai ʻona i hoʻokomo ʻia i loko o ka intravenous hiki ke hopena i ka hoʻonui nui ʻana o ke kaomi. Ua hōʻoia ʻia ʻo Fructus Aurantii a me Fructus Aurantii Fructus mai ʻekolu mau wahi noho like ʻole he mau hopena vasoconstriction iki e ka perfusion vascular o ke kino holoʻokoʻa o nā toads. I nā ʻīlio i hoʻomaʻemaʻe ʻia, aia kahi hopena hypertensive koʻikoʻi a wikiwiki. ʻAʻohe kaumaha hanu a i ʻole hypotension i hoʻokumu ʻia e ka epinephrine, a ʻaʻohe piʻi maopopo o ka helu o ka puʻuwai.
Pili ka ʻōnaehana hoʻonui kaomi i nā kumu aʻe:
3.1. Ka hoʻonāukiuki ʻana o nā mea loaʻa α, e hana ana i ka vasoconstriction i kekahi mau ʻōpū (hiki i ka phenylzoline ke hoʻohuli i ka hoʻonui ʻia o ke kaomi i loko o kahi hopena antihypertensive).
3.2. Hoʻonui ʻia ka ʻūlū ʻana o ka myocardial a me ka hoʻonui ʻana i ka puka cardiac (ka hoʻokaʻawale ʻana o ka perfusion puʻuwai guinea pig a me ka hoʻomākaukau cardiopulmonary). Ma hope o ka reserpine, ʻoi aku ka nui o ka hopena hoʻonui kaomi o Fructus aurantii aurantii. Ua hoʻonui nui ia i ke kahe o ke aʻa coronary (289.4% i hoʻonui ʻia ke kahe o ke aʻa coronary e ka bubble flowmeter) a hoʻonui i ke kahe o ke koko o ka lolo a me nā puʻupaʻa ma 86.4% a me 64.5% ma ka awelika, he ʻokoʻa loa ia mai ka norepinephrine. Aia ka emi ʻana o ke kahe koko femoral a me ka piʻi iki akā ʻaʻole nui i ka hoʻohana ʻana i ka oxygen myocardial, ʻaʻole i kūlike me ka hoʻonui nui ʻana o ke kahe coronary. I nā hoʻokolohua ECG i nā ʻīlio a me nā puaʻa guinea, ʻaʻole koʻikoʻi ka arrhythmia (ventricular tachycardia a i ʻole ka atrioventricular block) i hoʻokumu ʻia e kahi nui o ka aurantii aurantii. Ma muli o nā ʻano i luna, ua manaʻo ʻia e mālama i ka haʻalulu cardiogenic. Hiki i nā Alkaloids i hoʻokaʻawale ʻia mai Fructus Aurantii a me Lycium orange ke hoʻonui i ka ʻeha o ka ʻiʻo laumania vascular, ʻoiai ke mālama ʻia me ka pituitrin.
4. Antithrombotic: Ua hōʻike ka hoʻāʻo in vitro o 0.1g/ml Fructus Aurantii aqua decoction i kahi hopena antithrombotic maopopo.
5. Ka hopena anti-allergic: ʻO ka hoʻokomo ʻana o ka pulse static 100mg/kg o ka wai Fructus Aurantii Aurantii hiki ke kāohi i ka hopena maʻi ʻili passive (PCA) i loko o nā ʻiole, a hiki i ka 50μg/ml ke kāohi i ka hoʻokuʻu ʻana o ka histamine mai nā pūnaewele mast ʻōpū o ka ʻiole.
6. Nā hopena ʻē aʻe: Hiki i ka mycin o ka mea kanu citrus ke hōʻemi i ka nui o ka cholestatin i loko o ke serum a me ke akepaʻa o nā ʻiole i hānai ʻia me ka ʻai i loaʻa ka cholesterol. ʻO ka wai ʻona o Fructus Aurantii he hopena pale i ka mycobacterium tuberculosis H37Rv in vitro, a ʻo kona ʻano pale he 1:1000. ʻAʻohe hopena o kāna wai hoʻoheheʻe i ka bronchus guinea pig. Ua hōʻike ʻia ua hoʻonui ka wai hua citrus i ka wikiwiki o ka fermentation o ka hū a ʻaʻole e hōʻemi i kāna hana ma hope o ka hoʻolapalapa ʻana, no laila ʻaʻole ia he ʻāpana enzymatic. ʻO ka hoʻohana lapaʻau nui o ka wai ʻalani, ʻo ia ka waiwai i ka huaora C a loaʻa ka nui o nā huaora A a me B. ʻAʻohe huaora C o ka ʻili akā waiwai i ka huaora A. He ʻawaʻawa kona ʻono a hiki ke hoʻoikaika i ka ʻōpū. ʻO nā keiki e like me ka lawe ʻana i ka nui o nā ʻili hiki ke hoʻoulu i ka lāʻau make (ʻeha ʻōpū, cramps).
Kuhikuhi:http://www.a-hospital.com
NoʻO ka ʻāpana Citrus Aurantium, e ʻoluʻolu e hoʻokaʻaʻike mai iā mākou. Ke kali nei mākou iā ʻoe ma ʻaneʻi i kēlā me kēia manawa!!!
Ka manawa hoʻouna: Dec-15-2022



